成果/Result
- C11 , a novel fibroblast growth factor receptor 1 (FGFR1) inhibitor, suppresses breast cancer metastasis and angiogenesis被引量:3收藏
- 作者:Zhuo Chen Lin-jiang Tong Bai-you Tang Hong-yan Liu Xin Wang Tao Zhang Xian-wen Cao Yi Chen Hong-lin Li Xu-hong Qian Yu-fang Xu Hua Xie Jian Ding
- 机构:Division of Antitumor Pharmacology;Shanghai Key Laboratory of New Drug Design
- 来源:中国药理学报(英文版) 2019
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- 类呋喃香豆素的合成与DNA的结合及细胞毒性研究被引量:1收藏
- 作者:解丽娟 陈卓
- 机构:华侨大学生物医学学院;华东理工大学药学院
- 来源:《光谱学与光谱分析》 2014
- 关键词:呋喃香豆素 “最小嵌入” 类呋喃香豆素 DNA 抗肿瘤
- 摘要:呋喃香豆素类化合物无紫外光辅助照射时抗肿瘤活性低,为提高其正常情况下的抗肿瘤活性,依据"最小嵌入"假说对其进行结构改造。把呋喃香豆素结构中的呋喃环拆分出来,使其与香豆素由原来稠环相并的结合方式转变为通过化学键相连,得到合...
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- Naphthalimides and analogues as antitumor agents:A review on molecular design, bioactivity and mechanism of action被引量:0收藏
- 作者:Zhuo Chen Yufang Xu Xuhong Qian
- 机构:State Key Laboratory of Bioreactor Engineering
- 来源:中国化学快报(英文版) 2018
- 关键词:Naphthalimides Antitumor Structure activity relationship Drug design strategy Mechanism of action
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- Design,synthesis and biological evaluation of fluorescent derivatives of ursolic acid in living cells被引量:0收藏
- 作者:Wenyi Mei Lijuan Xie Xiaodong Zhang Cunjian Shi Fengzhi Wang Qiqi Fu Zhenjiang Zhao Honglin Li Yufang Xu Zhuo Chen
- 机构:Shanghai Key Laboratory of New Drug Design;Innovation Center for AI and Drug Discovery;Lingang Laboratory
- 来源:中国化学快报(英文版) 2024
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- Novel seven-membered ring-fused naphthalimide derivatives with potentials for cancer theranostics被引量:0收藏
- 作者:Yonghui Yang Xiayu Shi Zhuo Chen Yufang Xu Xuhong Qian Weiping Zhu
- 机构:State Key Laboratory of Bioreactor Engineering
- 来源:中国化学快报(英文版) 2023
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