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Antiproliferative and apoptosis-inducing activities of novel naphthalimide-cyclam conjugates through dual topoisomerase (topo) I/II inhibition被引量:31收藏 分享
作者:Tan, Shaoying Sun, Deheng Lyu, Jiankun Sun, Xiao Wu, Fangshu Li, Qiang Yang, Yiqi Liu, Jianxu Wang, Xin Chen, Zhuo Li, Honglin Qian, Xuhong Xu, Yufang
机构:E China Univ Sci & Technol
来源:BIOORGANIC & MEDICINAL CHEMISTRY  2015
关键词:Naphthalimide-cyclam conjugates   Antitumor agents   Topoisomerase I   Topoisomerase II   DNA intercalation   Apoptosis  
Novel metal complexes of naphthalimide-cyclam conjugates as potential multi-target receptor tyrosine kinase (RTK) inhibitors: Synthesis and biological evaluation被引量:20收藏 分享
作者:Tan, Shaoying Han, Kun Li, Qiang Tong, Linjiang Yang, Yiqi Chen, Zhuo Xie, Hua Ding, Jian Qian, Xuhong Xu, Yufang
机构:E China Univ Sci & Technol;Chinese Acad Sci
来源:EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY  2014
关键词:Metal complexes   Naphthalimide   Cyclam   RTK inhibitors   Antiproliferation   Antiangiogenesis  
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