文献类型：期刊文献

英文题名：A simple and efficient synthesis of fused morpholine pyrrolidines/piperdines with potential insecticidal activities

作者：Wang, Jiayi[1];Xu, Beiling[1];Si, Shanyu[1];Li, Hui[1];Song, Gonghua[1]

机构：[1]E China Univ Sci & Technol, Sch Pharm, Shanghai Key Lab Chem Biol, Shanghai 200237, Peoples R China

年份：2014

卷号：18

期号：4

起止页码：887

外文期刊名：MOLECULAR DIVERSITY

收录：;WOS:【SCI-EXPANDED(收录号:WOS:000343605000018)】；

基金：Financial support for this work from National Basic Research Program of China (973 Program) (Grant 2010CB126101) and National Natural Science Foundation of China (Grant 20972052) are gratefully acknowledged.

语种：英文

外文关键词：Multicomponent; Petasis-borono Mannich reaction; Fused morpholines; Insecticidal activity; MCR

摘要：A simple and efficient synthesis of fused morpholine pyrrolidine/piperdine core structures was accomplished via a Petasis-borono Mannich reaction of cyclic amino alcohols, glyoxal and arylboronic acids with moderate to good yields. The bioassay data showed that the synthesized compounds displayed selective insecticidal activities against armyworm and root-knot nematode.