文献类型：期刊文献

中文题名：Synthesis and Insecticidal Evaluation of Novel Phthalic Diamides Containing 1,2,3-Triazoles via Click Reaction

作者：Yinbo Chen[1];Youxin Xiao[1];Xusheng Shao[1];Xiaoyong Xu[1];Zhong Li[1]

机构：[1]Shanghai Key Laboratory of Chemical Biology,School of Pharmacy,East China University of Science and Technology,Shanghai 200237,China

年份：2014

卷号：32

期号：7

起止页码：592

中文期刊名：Chinese Journal of Chemistry

外文期刊名：中国化学（英文版）

收录：CSTPCD;;Scopus;CSCD:【CSCD2013_2014】；PubMed;

基金：This work was financially supported by the National Basic Research Program of China(973 Program,No.2010CB126100);the National High Technology Research and Development Program of China(863 Program Program,No.2011AA10A207);the National Natural Science Foundation of China(Nos.21372079;21272071);This work was also partly supported by the National Key Technology R&D Program of China(No.2011BAE06B01)and the Fundamental Research Funds for the Central Universities.

语种：英文

中文关键词：phthalic diamide;1,2,3-triazole;click chemistry;synthesis;bioactivity

摘要：A series of novel phthalic diamide derivatives containing 1,2,3-triazole moiety were synthesized using one-pot click chemistry approach and characterized by ^(1)H NMR and HRMS.The insecticidal activity against armyworm(Mythimna separata),Tetranychus cinnabarinus and cowpea aphid(Aphis craccivora)was evaluated.Compounds 4Ⅱ-a and 4Ⅱ-i showed 50%insecticidal activity against armyworm(Mythimna separata)at the concentration of 4 mg/L and one-third of the compounds had moderate activity against Tetranychus cinnabarinus at 500 mg/L.