文献类型：专利

英文题名：New isoxazole-3,5-bis(carboximidamide)compound useful in inhibiting pests or preventing pests and for preparing insecticidal composition

作者：LI Z;SHAO X;LEI C;XU X;CHENG J

机构：[1]UNIV EAST CHINA SCI & TECHNOLOGY

申请号：CN106632300-A

申请日：2016-09-29

公开日：2017-05-10

语种：英文

收录：DERWENT

摘要：NOVELTY - Isoxazole-3,5-bis(carboximidamide)compound (I) or salt are new. USE - (I) are useful in inhibiting pests or preventing pests and for preparing insecticidal composition (claimed). DETAILED DESCRIPTION - Isoxazole-3,5-bis(carboximidamide)compound of formula (I) or salt are new. R1 = H, 1-6C alkyl, allyl, 1-4C alkoxy-1-4C alkyl, 2-6C alkynyl-carbonyl, 2-3C alkenyl-carbonyl, 3-6C cycloalkyl-carbonyl, optionally substituted nitrogen, oxygen and/or sulfur of 5-6 membered heterocyclyl group, optionally substituted phenyl, optionally substituted benzyl, optionally substituted benzoyl or furanylcarbonyl; substituent = halo, 1-4C alkyl, 1-4C alkoxy, 1-4C haloalkyl, nitro, cyano or 1-4C haloalkoxy; either R2 and R3 = H, 1-6C alkyl, allyl, benzyl, 1-4C alkoxy-1-4C alkyl, 2-6C alkynyl-carbonyl, 2-3C alkenyl-carbonyl, 3-6C cycloalkyl-carbonyl, benzoyl, or substituted with halo, 1-4C alkyl group, 1-4C haloalkyl, 1-4C alkoxy, 1-4C haloalkoxy and 1-4C alkyl-carbonyl substituted with benzoyl, furanyl or N,N-dimethylcarbonyl; or R2 and R3 = together form -CH2-(CH2)n-CH2- ,-CH2-XR-CH2, -CH2-CH2-, -CH2-CH2-CH2- or -CH2-MRa-CH2-; M = N, O or S; Ra = absent or H, 1-6C alkyl or 1-4C alkoxy; n = 0-2; X = O, N or S; R = absent or H, 1-6C alkyl, allyl, benzyl, phenyl, 1-4C alkoxy-1-4C alkyl, 2-6C alkynyl-carbonyl, 2-3C alkenyl-carbonyl, 3-6C cycloalkyl-carbonyl, benzoyl or substituted with halo, 1-4C haloalkyl, 1-8C alkyl group or alkoxy group and 1-4C alkyl-carbonyl group, benzoyl group, furanyl group or N,N-dimethylcarbonyl; R4 = H, 1-6C alkyl, allyl, 1-4C alkoxy-1-4C alkyl, 2-6C alkynyl-carbonyl, 2-3C alkenyl-carbonyl, 3-6C cycloalkyl-carbonyl, optionally substituted nitrogen, oxygen and/or sulfur of five- or six-membered heterocyclic group, optionally substituted phenyl, optionally substituted benzyl, optionally substituted benzoyl group, furanyl carbonyl, optionally substituted nitrogen, oxygen and/or sulfur of 5-6 membered heterocyclic methyl; and substituent = halo, 1-4C alkyl, 1-4C alkoxy, 1-4C haloalkyl or 1-4C haloalkoxy. INDEPENDENT CLAIMS are also included for: (1) preparation of (I); and (2) agricultural composition comprising (i) 0.001-99.99 wt.% (I) or salt and (ii) carrier and/or excipient; (3) use of (I) comprising (i) inhibiting pests or preventing pests, (ii) preparing insecticidal composition; and (4) insecticidal and/or pest controlling method comprising reacting (I) or salt or agricultural composition, applying to plant, animal suffering from pests and its surrounding soil under environment.