- Discovery and Rational Design of Natural-Product-Derived 2-Phenyl-3,4-dihydro-2H-benzo[f]chromen-3-amine Analogs as Novel and Potent Dipeptidyl Peptidase 4 (DPP-4) Inhibitors for the Treatment of Type 2 Diabetes被引量:51收藏
- 作者:Li, Shiliang Xu, Hongling Cui, Shichao Wu, Fangshu Zhang, Youli Su, Mingbo Gong, Yinghui Qiu, Shaobing Jiao, Qian Qin, Chun Shan, Jiwei Zhang, Ming Wang, Jiawei Yin, Qiao Xu, Minghao Liu, Xiaofeng Wang, Rui Zhu, Lili Li, Jia Xu, Yufang Jiang, Hualiang Zhao, Zhenjiang Li, Jingya Li, Honglin
- 机构:East China Univ Sci & Technol;Chinese Acad Sci
- 来源:JOURNAL OF MEDICINAL CHEMISTRY 2016
- 质疑
- α-Functionalization of 2-Vinylpyridines via a Chiral Phosphine Catalyzed Enantioselective Cross Rauhut-Currier Reaction被引量:42收藏
- 作者:Qin, Cong Liu, Yonghai Yu, Yang Fu, Yiwei Li, Hao Wang, Wei
- 机构:East China Univ Sci & Technol;East China Univ Sci & Technol;Univ New Mexico
- 来源:ORGANIC LETTERS 2018
- 质疑
- Co(OAc)2-Catalyzed Trifluoromethylation and C(3)-Selective Arylation of 2-(Propargylamino)pyridines via a 6-Endo-Dig Cyclization被引量:37收藏
- 作者:Li, Jianjun Lei, Yifan Yu, Yang Qin, Cong Fu, Yiwei Li, Hao Wang, Wei
- 机构:East China Univ Sci & Technol;East China Univ Sci & Technol;Univ New Mexico
- 来源:ORGANIC LETTERS 2017
- 质疑
- Discovery of a Natural-Product-Derived Preclinical Candidate for Once-Weekly Treatment of Type 2 Diabetes被引量:29收藏
- 作者:Li, Shiliang Qin, Chun Cui, Shichao Xu, Hongling Wu, Fangshu Wang, Jiawei Su, Mingbo Fang, Xiaoyu Li, Dan Jiao, Qian Zhang, Ming Xia, Chunmei Zhu, Lili Wang, Rui Li, Jia Jiang, Hualiang Zhao, Zhenjiang Li, Jingya Li, Honglin
- 机构:East China Univ Sci & Technol;Chinese Acad Sci;Univ Chinese Acad Sci
- 来源:JOURNAL OF MEDICINAL CHEMISTRY 2019
- 质疑
- Lewis Acid-Catalyzed C(sp3)-C(sp3) Bond Forming Cyclization Reactions for the Synthesis of Tetrahydroprotoberberine Derivatives被引量:22收藏
- 作者:Li, Jianjun Qin, Cong Yu, Yang Fan, Huaqiang Fu, Yiwei Li, Hao Wang, Wei
- 机构:East China Univ Sci & Technol;East China Univ Sci & Technol;Univ New Mexico
- 来源:ADVANCED SYNTHESIS & CATALYSIS 2017
- 关键词:annulation azaarene activation C(sp(3))-C(sp(3)) bond formation Lewis acid catalysis tetrahydroprotoberberine derivatives
- 质疑
- Asymmetric synthesis of isoquinolinonaphthyridines catalyzed by a chiral Bronsted acid被引量:22收藏
- 作者:Li, Jianjun Fu, Yiwei Qin, Cong Yu, Yang Li, Hao Wang, Wei
- 机构:East China Univ Sci & Technol;East China Univ Sci & Technol;Univ New Mexico
- 来源:ORGANIC & BIOMOLECULAR CHEMISTRY 2017
- 质疑
- Alkenylazaarenes as dipolarophiles in 1,3-dipolar cycloaddition of nitrones: regioselectivity-switchable and highly diastereoselective synthesis of multisubstituted isoxazolidines被引量:16收藏
- 作者:Tong, Mengchao Zhang, Yong Qin, Cong Fu, Yiwei Liu, Yonghai Li, Hao Wang, Wei
- 机构:East China Univ Sci & Technol;East China Univ Sci & Technol;Univ New Mexico
- 来源:ORGANIC CHEMISTRY FRONTIERS 2018
- 关键词:Microwave irradiation - Stereoselectivity
- 质疑
- Direct Access of the Chiral Quinolinyl Core of Cinchona Alkaloids via a Bronsted Acid and Chiral Amine Co-catalyzed Chemo- and Enantioselective α-Alkylation of Quinolinylmethanols with Enals被引量:9收藏
- 作者:Tong, Mengchao Wang, Sinan Zhuang, Jinchen Qin, Cong Li, Hao Wang, Wei
- 机构:East China Univ Sci & Technol;East China Univ Sci & Technol;Univ New Mexico
- 来源:ORGANIC LETTERS 2018
- 质疑
- Iron-Catalyzed Anti-Markovnikov Hydroamination of Vinylpyridines被引量:7收藏
- 作者:Peng, Yahui Qin, Cong Chen, Xiaobei Li, Jianjun Li, Hao Wang, Wei
- 机构:East China Univ Sci & Technol;East China Univ Sci & Technol;Univ New Mexico
- 来源:ASIAN JOURNAL OF ORGANIC CHEMISTRY 2017
- 关键词:anti-Markovnikov azoles hydroamination iron vinylpyridines
- 质疑
- A Facile Oxidation of Tertiary Amines to Lactams by Using Sodium Chlorite: Process Improvement by Precise pH Adjustment with CO2被引量:6收藏
- 作者:Liu, Chaoyang Sun, Haozhou Qin, Cheng Yang, Tiannuo Zhang, Wenxian Zhou, Yuan Li, Yani Jia, Zheng Robert Chu, Changhu
- 机构:East China Univ Sci & Technol;East China Univ Sci & Technol;East China Univ Sci & Technol;Shanghai High Sch
- 来源:SYNLETT 2022
- 关键词:amine oxidation sodium chlorite transition-metal-free carbon dioxide pH adjustment
- 质疑
- [4+2] Cycloaddition of trifluoromethyl ketimines with 2-alkenyl azaarenes through selective C-F bond cleavage of CF3被引量:6收藏
- 作者:Fu, Yiwei Qin, Cong Zhang, Zhiqiang Shi, Haoyu Zhao, Jianbo Gong, Xueqing Shi, Lei Li, Hao
- 机构:East China Univ Sci & Technol;East China Univ Sci & Technol;East China Univ Sci & Technol;East China Univ Sci & Technol;East China Univ Sci & Technol
- 来源:ORGANIC CHEMISTRY FRONTIERS 2021
- 质疑
- Facile Preparation of 4-(4-Nitrophenyl)morpholin-3-one via the Acid-Catalyzed Selective Oxidation of 4-(4-Nitrophenyl)morpholine by Sodium Chlorite as the Sole Oxidant被引量:5收藏
- 作者:Liu, Chaoyang Yu, Tao Yang, Tiannuo Sun, Haozhou Qin, Cheng Jia, Qiang Chu, Changhu
- 机构:East China Univ Sci & Technol;East China Univ Sci & Technol;Seasons Biotechnol Taizhou Co Ltd
- 来源:ORGANIC PROCESS RESEARCH & DEVELOPMENT 2020
- 关键词:rivaroxaban 4-(4-nitrophenyl)morpholin-3-one oxidation sodium chlorite
- 质疑
- Water-based DNF@PLA microcapsules with excellent interface properties enhancing insecticidal activity against Nilaparvata lugens被引量:0收藏
- 作者:Qin, Chen Gao, Yue Zhang, Bo Zhou, Cong Sun, Li Zou, Aihua Cheng, Jiagao
- 机构:East China Univ Sci & Technol;Shanghai Normal Univ;East China Univ Sci & Technol
- 来源:PEST MANAGEMENT SCIENCE 2026
- 关键词:dinotefuran insecticidal activity interfacial properties microcapsules W/O emulsion
- 质疑
- Extending the concentration limit of electrodialytic eluent generator for ion chromatography被引量:0收藏
- 作者:Chen, Weiqing Jin, Huiling Qin, Cheng Zhang, Feifang Yang, Bingcheng
- 机构:East China Univ Sci & Technol
- 来源:TALANTA 2027
- 关键词:Ion chromatography Electrodialytic eluent generator Dual-membrane Single-membrane Concentration limit Gas-free
- 质疑


