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  • 人物=李忠 x

502 条 记 录,以下是 1-30

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Divalent and Oxabridged Neonicotinoids Constructed by Dialdehydes and Nitromethylene Analogues of Imidacloprid: Design, Synthesis, Crystal Structure, and Insecticidal Activities被引量:116收藏 分享
作者:Shao, Xusheng Fu, Hua Xu, Xiaoyong Xu, Xinglei Liu, Zewen Li, Zhong Qian, Xuhong
机构:E China Univ Sci & Technol;Nanjing Agr Univ;Qinghai Univ
来源:JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY  2010
关键词:Neonicotinoids   dialdehydes   imidacloprid   insecticide   oxabridge  
Overall status of neonicotinoid insecticides in China: Production, application and innovation被引量:112收藏 分享
作者:Shao, Xusheng Liu, Zewen Xu, Xiaoyong Li, Zhong Qian, Xuhong
机构:E China Univ Sci & Technol;Nanjing Agr Univ
来源:JOURNAL OF PESTICIDE SCIENCE  2013
关键词:China   neonicotinoid   production   application   innovation  
Synthesis, insecticidal activity, and QSAR of novel nitromethylene neonicotinoids with tetrahydropyridine fixed cis configuration and exo-ring ether modification被引量:107收藏 分享
作者:Tian, Zhongzhen Shao, Xusheng Li, Zhong Qian, Xuhong Huang, Qingchun
机构:E China Univ Sci & Technol
来源:JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY  2007
关键词:nitromethylene   tetrahydropyridine   cis position   QSAR  
Novel 1,3,4-Oxadiazole-2-carbohydrazides as Prospective Agricultural Antifungal Agents Potentially Targeting Succinate Dehydrogenase被引量:105收藏 分享
作者:Wu, Yuan-Yuan Shao, Wu-Bin Zhu, Jian-Jun Long, Zhou-Qing Liu, Li-Wei Wang, Pei-Yi Li, Zhong Yang, Song
机构:Guizhou Univ;East China Univ Sci & Technol
来源:JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY  2019
关键词:1,3,4-oxadiazole   carbohydrazide   bioactivity   succinate dehydrogenase inhibitor  
Design, Synthesis, and Insecticidal Activities of Novel Analogues of Neonicotinoids: Replacement of Nitromethylene with Nitroconjugated System被引量:75收藏 分享
作者:Shao, Xusheng Li, Zhong Qian, Xuhong Xu, Xiaoyong
机构:E China Univ Sci & Technol
来源:JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY  2009
关键词:Neonicotinoids   nitromethylene   imidacloprid   insecticide  
Rational Optimization and Action Mechanism of Novel Imidazole (or Imidazolium)-Labeled 1,3,4-Oxadiazole Thioethers as Promising Antibacterial Agents against Plant Bacterial Diseases被引量:75收藏 分享
作者:Wang, Pei-Yi Wang, Ming-Wei Zeng, Dan Xiang, Meng Rao, Jia-Rui Liu, Qing-Qing Liu, Li -Wei Wu, Zhi-Bing Li, Zhong Song, Bao-An Yang, Song
机构:Guizhou Univ;East China Univ Sci & Technol
来源:JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY  2019
关键词:1,3,4-oxadiazole   imidazole or imidazolium   antibacterial   action mechanism  
cis-Nitromethylene neonicotinoids as new nicotinic family: Synthesis, structural diversity, and insecticidal evaluation of hexahydroimidazo[1,2-α]pyridine被引量:75收藏 分享
作者:Shao, Xusheng Zhang, Wenwen Peng, Yanqing Li, Zhong Tian, Zhongzhen Qian, Xuhong
机构:E China Univ Sci & Technol
来源:BIOORGANIC & MEDICINAL CHEMISTRY LETTERS  2008
关键词:Neonicotinoid   cis-Configuration   Insecticide   Resistance  
Designing Tetrahydroimidazo[1,2-a]pyridine Derivatives via Catalyst-free Aza-Diels-Alder Reaction (ADAR) and Their Insecticidal Evaluation被引量:70收藏 分享
作者:Zhang, Wenwen Chen, Yinbo Chen, Weidong Liu, Zewen Li, Zhong
机构:E China Univ Sci & Technol;Nanjing Agr Univ
来源:JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY  2010
关键词:Aza-Diels-Alder   catalyst-free   insecticide   biological activities  
cis-Configuration: A New Tactic/Rationale for Neonicotinoid Molecular Design被引量:70收藏 分享
作者:Shao, Xusheng Lee, Philip W. Liu, Zewen Xu, Xiaoyong Li, Zhong Qian, Xuhong
机构:E China Univ Sci & Technol;Nanjing Agr Univ
来源:JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY  2011
关键词:neonicotinoids   cis-configuration   insecticide   selectivity  
害虫对新烟碱类杀虫剂的抗药性及其治理策略被引量:69收藏 分享
作者:唐振华 陶黎明 李忠
机构:华东理工大学药学院;上海农药研究所
来源:《农药学学报》  2006
关键词:新烟碱类杀虫剂  抗性机理  P450单加氧酶  靶标部位抗性  抗性治理  
摘要:烟碱和新烟碱类杀虫剂都是作为后突触烟碱乙酰胆碱受体(nAChRs)的激动剂作用于昆虫中枢神经系统,但这两类杀虫剂存在明显不同的选择毒性:烟碱类对哺乳动物毒性较高,而杀虫活性低;新烟碱类具有高杀虫活性,而对哺乳动物低毒。由...
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Antibacterial Functions and Proposed Modes of Action of Novel 1,2,3,4-Tetrahydro-β-carboline Derivatives that Possess an Attractive 1,3-Diaminopropan-2-ol Pattern against Rice Bacterial Blight, Kiwifruit Bacterial Canker, and Citrus Bacterial Canker被引量:68收藏 分享
作者:Liu, Hong-Wu Ji, Qing-Tian Ren, Gang-Gang Wang, Fang Su, Fen Wang, Pei-Yi Zhou, Xiang Wu, Zhi-Bing Li, Zhong Yang, Song
机构:Guizhou Univ;East China Univ Sci & Technol
来源:JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY  2020
关键词:tetrahydro-beta-carboline derivatives   antiphytopathogen   in vitro and in vivo bioassays   ROS   apoptosis   hypersensitive response  
Pyrrole- and Dihydropyrrole-Fused Neonicotinoids: Design, Synthesis, and Insecticidal Evaluation被引量:64收藏 分享
作者:Ye, Zhenjun Shi, Lina Shao, Xusheng Xu, Xiaoyong Xu, Zhiping Li, Zhong
机构:E China Univ Sci & Technol
来源:JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY  2013
关键词:Pyrrole   dihydropyrrole   neonicotinoid   nAChR  
Synthesis and In Vitro and In Vivo Biological Activity Evaluation and Quantitative Proteome Profiling of Oxadiazoles Bearing Flexible Heterocyclic Patterns被引量:63收藏 分享
作者:Tao, Qing-Qing Liu, Li-Wei Wang, Pei-Yi Long, Qing-Su Zhao, Yong-Liang Jin, Lin-Hong Xu, Wei-Ming Chen, Yang Li, Zhong Yang, Song
机构:Guizhou Univ;East China Univ Sci & Technol
来源:JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY  2019
关键词:oxadiazoles   heterocyclic patterns   biological activity   quantitative proteomics  
Identification of Racemic and Chiral Carbazole Derivatives Containing an Isopropanolamine Linker as Prospective Surrogates against Plant Pathogenic Bacteria: In Vitro and In Vivo Assays and Quantitative Proteomics被引量:62收藏 分享
作者:Zhao, Yong-Lian Huang, Xing Liu, Li-Wei Wang, Pei-Yi Long, Qing-Su Tao, Qing-Qing Li, Zhong Yang, Song
机构:Guizhou Univ;East China Univ Sci & Technol
来源:JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY  2019
关键词:carbazole   isopropanolamine   antibacterial   proteomics   action mechanism  
Selenium-containing naphthalimides as anticancer agents: Design, synthesis and bioactivity被引量:60收藏 分享
作者:Zhao, Liwei Li, Jianfeng Li, Yiquan Liu, Jianwen Wirth, Thomas Li, Zhong
机构:E China Univ Sci & Technol;Cardiff Univ
来源:BIOORGANIC & MEDICINAL CHEMISTRY  2012
关键词:Anticancer   Naphthalimides   Selenium   K562   DNA  
Characterization of hepatotoxic effects induced by pyraclostrobin in human HepG2 cells and zebrafish larvae被引量:60收藏 分享
作者:Wu, Mengqi Bian, Jinhao Han, Shuang Zhang, Cheng Xu, Wenping Tao, Liming Li, Zhong Zhang, Yang
机构: Shanghai Key Laboratory of Chemical Biology; Department of Pathology; State Key Laboratory of Bioreactor Engineering
来源:Chemosphere  2023
关键词:Activation analysis - Disease control - Mitochondria  
Synthesis of Thiazolium-Labeled 1,3,4-Oxadiazole Thioethers as Prospective Antimicrobials: In Vitro and in Vivo Bioactivity and Mechanism of Action被引量:59收藏 分享
作者:Wang, Ming-Wei Zhu, Huai-He Wang, Pei-Yi Zeng, Dan Wu, Yuan-Yuan Liu, Li-Wei Wu, Zhi-Bing Li, Zhong Yang, Song
机构:Guizhou Univ;East China Univ Sci & Technol
来源:JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY  2019
关键词:1,3,4-oxadiazole   thiazolium   antimicrobial   3D-QSAR   proteomics   action mechanism  
Developmental toxicity and estrogenicity of glyphosate in zebrafish in vivo and in silico studies被引量:58收藏 分享
作者:Lu, Jian Zhang, Cheng Xu, Wenping Chen, Weidong Tao, Liming Li, Zhong Cheng, Jiagao Zhang, Yang
机构: Shanghai Key Laboratory of Chemical Biology; Department of Pathology
来源:Chemosphere  2023
关键词:Animals - Deep learning - Endocrine disrupters - Herbicides  
Surface Morphology and the Action Mechanism of Macrophage Immuno-Stimulating Activity of Rosa Setate X Rosa Rugosa Polysaccharide Wsrp-1b被引量:57收藏 分享
作者:Wu, Mengqi Xu, Jingying Li, Wei Han, Qifeng Xia, Wei Li, Zhong Zhang, Yang Zhang, Wenqing
机构: Shanghai Key Laboratory of Chemical Biology; Shanghai Key Laboratory of Functional Materials Chemistry; State Key Laboratory of Dairy Biotechnology
来源:SSRN  2023
关键词:Antigen-antibody reactions - Azo dyes - Disease control - Electrophoresis - Morphology - Nitric oxide - Scanning electron microscopy - Surface morphology  
Synthesis and Nematicidal Activities of 1,2,3-Benzotriazin-4-one Derivatives against Meloidogyne incognita被引量:57收藏 分享
作者:Wang, Gaolei Chen, Xiulei Deng, Yayun Li, Zhong Xu, Xiaoyong
机构:E China Univ Sci & Technol;Shanghai Collaborat Innovat Ctr Biomfg Technol
来源:JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY  2015
关键词:1,2,3-benzotriazin-4-one   2-cyanoiminothiazolidin-4-one   nematicide   Meloidogyne incognita   in vivo  
The thiazoylmethoxy modification on pyrazole oximes: Synthesis and insecticidal biological evaluation beyond acaricidal activity被引量:56收藏 分享
作者:Dai, Hong Xiao, Yan-Shuang Li, Zhong Xu, Xiao-Yong Qian, Xu-Hong
机构:E China Univ Sci & Technol;Nantong Univ
来源:CHINESE CHEMICAL LETTERS  2014
关键词:Pyrazole oxime   Substituted thiazole   Acaricidal activity   Insecticidal activity  
Characterization of glyphosate-induced cardiovascular toxicity and apoptosis in zebrafish被引量:55收藏 分享
作者:Lu, Jian Wang, Weiguo Zhang, Cheng Xu, Wenping Chen, Weidong Tao, Liming Li, Zhong Cheng, Jiagao Zhang, Yang
机构:East China Univ Sci & Technol;UT southwestern Med Ctr
来源:SCIENCE OF THE TOTAL ENVIRONMENT  2022
关键词:Glyphosate   Developmental toxicity   Heart   Vascular   Apoptosis   Zebra fish  
Insights into pesticide toxicity against aquatic organism: QSTR models on Daphnia Magna被引量:53收藏 分享
作者:He, Lujue Xiao, Keya Zhou, Cong Li, Guanglong Yang, Hongbin Li, Zhong Cheng, Jiagao
机构:East China Univ Sci & Technol;East China Univ Sci & Technol
来源:ECOTOXICOLOGY AND ENVIRONMENTAL SAFETY  2019
关键词:Pesticide   Aquatic toxicity   Daphnia magna   Quantitative structure toxicity relationship (QSTR)   Machine learning  
Specific Synergist for Neonicotinoid Insecticides: IPPA08, a cis-Neonicotinoid Compound with a Unique Oxabridged Substructure被引量:53收藏 分享
作者:Bao, Haibo Shao, Xusheng Zhang, Yixi Deng, Yayun Xu, Xiaoyong Liu, Zewen Li, Zhong
机构:Nanjing Agr Univ;E China Univ Sci & Technol
来源:JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY  2016
关键词:neonicotinoid   insecticide synergist   detoxification enzyme   nicotinic acetylcholine receptors  
Cis-configuration: A new tactic/rationale for neonicotinoid molecular design被引量:52收藏 分享
作者:Shao, Xusheng Lee, Philip W. Liu, Zewen Xu, Xiaoyong Li, Zhong Qian, Xuhong
机构: Shanghai Key Laboratory of Chemical Biology; Key Laboratory of Monitoring and Management of Plant Disease and Insect
来源:Journal of Agricultural and Food Chemistry  2011
关键词:Organic compounds  
Simultaneous Quantification of Hg2+ and MeHg+ in Aqueous Media with a Single Fluorescent Probe by Multiplexing in the Time Domain被引量:51收藏 分享
作者:Zhang, Ziqian Zhang, Baoyan Qian, Xuhong Li, Zhong Xu, Zhiping Yang, Youjun
机构:E China Univ Sci & Technol;E China Univ Sci & Technol
来源:ANALYTICAL CHEMISTRY  2014
关键词:Cost effectiveness - Time domain analysis  
An unusual synthesis of Troger's bases using DMSO/HCl as formaldehyde equivalent被引量:50收藏 分享
作者:Li, Z Xu, XY Peng, YQ Jiang, ZX Ding, CY Qian, XH
机构:E China Univ Sci & Technol;Dalian Univ Technol
来源:SYNTHESIS-STUTTGART  2005
关键词:Troger's bases   DMSO/HCl   formaldehyde equivalent  
Synthesis and Docking Study of N-(Cinnamoyl)-N′-(substituted)acryloyl Hydrazide Derivatives Containing Pyridinium Moieties as a Novel Class of Filamentous Temperature-Sensitive Protein Z Inhibitors against the Intractable Xanthomonas oryzae pv. oryzae Infections in Rice被引量:50收藏 分享
作者:Zhou, Xiang Feng, Yu-Mei Qi, Pu-Ying Shao, Wu-Bin Wu, Zhi-Bing Liu, Li-Wei Wang, Yi Ma, Hao-Dong Wang, Pei-Yi Li, Zhong Yang, Song
机构:Guizhou Univ;East China Univ Sci & Technol
来源:JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY  2020
关键词:rice bacterial blight   diacylhydrazine derivatives   FtsZ inhibitor   antibacterial assay  
Actions between neonicotinoids and key residues of insect nAChR based on an ab initio quantum chemistry study:: Hydrogen bonding and cooperative π-π interaction被引量:50收藏 分享
作者:Wang, Yanli Cheng, Jiagao Qian, Xuhong Li, Zhong
机构:E China Univ Sci & Technol
来源:BIOORGANIC & MEDICINAL CHEMISTRY  2007
关键词:neonicotinoids   nicotinic acetylcholine receptor   binding model  
Characterization of Glyphosate-Induced Cardiovascular Toxicity and Apoptosis in Zebrafish Embryos被引量:49收藏 分享
作者:Lu, Jian Wang, Weiguo Zhang, Cheng Xu, Wenping Tao, Liming Li, Zhong Cheng, Jiagao Zhang, Yang
机构: Shanghai Key Laboratory of Chemical Biology; Department of Pathology
来源:SSRN  2022
关键词:Cell death - Health hazards - Herbicides  
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