付稳 收藏

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( 任职于 药学院药物化工研究所)

被引量:274H指数:9SCI-EXPANDED: 24 EI: 16 北大核心: 1 CSCD: 1

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33 条 记 录,以下是 1-30

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Rational Exploration of Novel SDHI Fungicide through an Amide-?-ketonitrile Bioisosteric Replacement Strategy被引量:42收藏 分享
作者:Zhou, Cong Sun, Xujuan Fu, Wen Li, Zhong Cheng, Jiagao Maienfisch, Peter
机构:East China Univ Sci & Technol
来源:JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY  2023
关键词:?-ketonitriles   succinate dehydrogenase inhibitors   fungicidal activity   bioisosteric replacement   molecular docking   3D-QSAR  
质疑
Application of photopharmacology in agrochemicals被引量:35收藏 分享
作者:Fu, Wen Li, Zhong Shao, Xusheng
机构:East China Univ Sci & Technol;East China Univ Sci & Technol;East China Univ Sci & Technol;East China Univ Sci & Technol
来源:ADVANCED AGROCHEM  2023
关键词:Photopharmacology   Agrochemicals   Photochromic ligands   Optical control   Ligand-receptor interactions  
质疑
Synthesis and Biological Activity of Novel Antifungal Leads: 3,5-Dichlorobenzyl Ester Derivatives被引量:29收藏 分享
作者:Du, Shaoqing Yuan, Qinglong Hu, Xueping Fu, Wen Xu, Qi Wei, Ziyi Xu, Jiazheng Shao, Xusheng Qian, Xuhong
机构:East China Univ Sci & Technol;Zhejiang Univ;East China Normal Univ
来源:JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY  2021
关键词:succinate dehydrogenase inhibitors   fungicidal activity   molecular dynamic simulations   3,5-dichlorobenzyl ester  
质疑
Reversible Regulation of Succinate Dehydrogenase by Tools of Photopharmacology被引量:28收藏 分享
作者:Fu, Wen Shao, Zhongli Sun, Xujuan Zhou, Cong Xu, Zhiping Zhang, Yang Cheng, Jiagao Li, Zhong Shao, Xusheng
机构:East China Univ Sci & Technol;East China Univ Sci & Technol;East China Univ Sci & Technol
来源:JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY  2022
关键词:regulation   SDH   photochromic ligands   azobenzene   optical control  
质疑
Azo-incorporating Increases Inhibitory Activity of Succinate Dehydrogenase被引量:26收藏 分享
作者:Fu, Wen Hu, Xinyue Yuan, Qinglong Sun, Xujuan Xu, Zhiping Zhang, Yang Cheng, Jiagao Ye, Yonghao Li, Zhong Shao, Xusheng
机构:East China Univ Sci & Technol;Nanjing Agr Univ;East China Univ Sci & Technol
来源:JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY  2021
关键词:azobenzene   activity   fungicide   succinate dehydrogenase  
质疑
Azobenzene-Semicarbazone Enables Optical Control of Insect Sodium Channels and Behavior被引量:17收藏 分享
作者:Qiao, Zhi Fu, Wen Zhang, Yongchao Chen, Ruijia Xu, Zhiping Li, Zhong Shao, Xusheng
机构:East China Univ Sci & Technol;East China Univ Sci & Technol
来源:JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY  2021
关键词:photopharmacology   sodium channels   photoswitches   metaflumizone   invertebrates  
质疑
Novel SDH Inhibitors as Antifungal Leads: From Azobenzene Derivatives to the 1,2,4-Oxadiazole Compounds被引量:14收藏 分享
作者:Fu, Wen Yuan, Qinglong Zhang, Hangji Li, Xiaoyan Lu, Yiming Yan, Wenming Ye, Yonghao Liu, Xili Li, Zhong Shao, Xusheng
机构:East China Univ Sci & Technol;Guizhou Univ;Yantai Inst China Agr Univ;Shandong Yingxin Chem Co Ltd;Nanjing Agr Univ
来源:JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY  2024
关键词:SDH   azobenzene   1,2,4-oxadiazole   antifungal lead   structural optimization  
质疑
Design, synthesis and bioassay of the emerging photo-responsive fungicides被引量:11收藏 分享
作者:Fu, Wen Hu, Xinyue Yuan, Qinglong Xu, Zhiping Cheng, Jiagao Li, Zhong Shao, Xusheng
机构:East China Univ Sci & Technol;East China Univ Sci & Technol;East China Univ Sci & Technol;East China Univ Sci & Technol
来源:CHINESE CHEMICAL LETTERS  2023
关键词:Phenamacril   Controlled release   Photoremovable protecting groups   Spatiotemporal   Significant difference  
质疑
The potential immunotoxicity of emamectin benzoate on the human THP-1 macrophages被引量:10收藏 分享
作者:Wei, Ziyi Wang, Weiguo Fu, Wen Zhang, Ping Feng, Hao Xu, Wenping Tao, Liming Li, Zhong Zhang, Yang Shao, Xusheng
机构:East China Univ Sci & Technol;East China Univ Sci & Technol;East China Univ Sci & Technol;East China Univ Sci & Technol
来源:ENVIRONMENTAL TOXICOLOGY  2023
关键词:emamectin benzoate   immunotoxicity   NF-kappa B pathway   pesticide   THP-1 macrophages  
质疑
Dual photo-controlled release system for fipronil and dinotefuran被引量:8收藏 分享
作者:Fu, Wen Du, Kang Xu, Zhiping Cheng, Jiagao Li, Zhong Shao, Xusheng
机构:East China Univ Sci & Technol;East China Univ Sci & Technol;East China Univ Sci & Technol;East China Univ Sci & Technol
来源:PHOTOCHEMICAL & PHOTOBIOLOGICAL SCIENCES  2023
关键词:Dual release   TNB-insecticides   Light   Synergistic effect   Pesticide delivery  
质疑
Optical Regulation of GABA Receptor by Visible Light via Azobenzene-Phenylpyrazole被引量:7收藏 分享
作者:Qiao, Zhi Fu, Wen Huang, Qiutang Li, Zhong Zhao, Chunqing Shao, Xusheng
机构:East China Univ Sci & Technol;Nanjing Agr Univ;East China Univ Sci & Technol;East China Univ Sci & Technol
来源:JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY  2022
关键词:photopharmacology   GABARs   azobenzene   phenylpyrazole   photoregulation  
质疑
Design, synthesis, and biological activity of heterocyclic methyl esters被引量:6收藏 分享
作者:Yuan, Qinglong Zhang, Yongchao Du, Shaoqing Fu, Wen Xu, Zhiping Cheng, Jiagao Li, Zhong Shao, Xusheng
机构:East China Univ Sci & Technol;Shandong Univ;East China Univ Sci & Technol;East China Univ Sci & Technol;East China Univ Sci & Technol
来源:JOURNAL OF HETEROCYCLIC CHEMISTRY  2023
质疑
Light Regulation of Insect Behavior by Azobenzene-modified Flonicamid as Novel Molecular Tools被引量:5收藏 分享
作者:Sheng, Zhubo Fu, Wen Zhang, Hangji Wang, Weiguo Li, Xiaoyan Xu, Zhiping Li, Zhong Shao, Xusheng
机构:East China Univ Sci & Technol;Guizhou Univ;China Agr Univ;East China Univ Sci & Technol;East China Univ Sci & Technol
来源:JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY  2024
关键词:photopharmacology   azobenzene   photoregulation   Naam   AlphaFold2  
质疑
Acid-promoted reaction of N-(cyanomethyl) amide with nitrosation reagent: Facile synthesis of 1,2,4-oxadiazole-3-carboxamide被引量:5收藏 分享
作者:Du, Shaoqing Li, Jin Fu, Wen Xu, Xiaoyong Shao, Xusheng Qian, Xuhong
机构:East China Univ Sci & Technol;East China Normal Univ
来源:TETRAHEDRON LETTERS  2021
关键词:N-(Cyanomethyl)amide   1   2   4-Oxadiazole-3-carboxamide   Methyl 1   2   4-oxadiazole-3-carboxylate   N0-Hydroxycarbamimidoyl cyanide  
质疑
Discovery of Novel Nicotinamide Derivatives by a Two-Step Strategy of Azo-Incorporating and Bioisosteric Replacement被引量:5收藏 分享
作者:Ru, Yifan Fu, Wen Guo, Sifan Li, Xiaoyan Zhou, Cong Xu, Zhiping Cheng, Jiagao Li, Zhong Shao, Xusheng
机构:East China Univ Sci & Technol;Yantai Inst China Agr Univ;East China Univ Sci & Technol
来源:JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY  2024
关键词:nicotinamide   azo-incorporating   bioisostericreplacement   fungicidal spectrum   SDH  
质疑
Application of TNB in dual photo-controlled release of phenamacril, imidacloprid, and imidacloprid synergist被引量:4收藏 分享
作者:Yin, Qi Fu, Wen Hu, Xinyue Xu, Zhiping Li, Zhong Shao, Xusheng
机构:East China Univ Sci & Technol;East China Univ Sci & Technol;East China Univ Sci & Technol;East China Univ Sci & Technol
来源:PHOTOCHEMISTRY AND PHOTOBIOLOGY  2024
关键词:dual photo-controlled release   fungicide   insecticide   synergist   TNB  
质疑
Optical Regulation of Sodium Channels by the Azobenzene Pyrethrins被引量:4收藏 分享
作者:Fu, Wen Ji, Yunfan Zhang, Yanan Xu, Jiazheng Xu, Zhiping Cheng, Jiagao Li, Zhong Shao, Xusheng
机构:East China Univ Sci & Technol;East China Normal Univ;East China Univ Sci & Technol;East China Univ Sci & Technol;East China Univ Sci & Technol
来源:ACS AGRICULTURAL SCIENCE & TECHNOLOGY  2022
关键词:azobenzene   pyrethrins   optical control   insecticidal activities   sodium channel  
质疑
Optical Control of Insect Behavior and Receptors with Azobenzene-Bridged Fipronil and Imidacloprid被引量:4收藏 分享
作者:Fu, Wen Sheng, Zhubo Qiao, Zhi Xu, Zhiping Li, Meng Guan, Ying Li, Zhong Shao, Xusheng
机构:East China Univ Sci & Technol;East China Univ Sci & Technol;East China Univ Sci & Technol;East China Univ Sci & Technol;Joint Inst Tobacco & Hlth
来源:JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY  2024
关键词:azobenzene bridge   multiphoton   insect receptorand behavior   spatiotemporal   regulation  
质疑
Enantioselective synthesis of 2-amino-4H-chromene derivatives with antifungal activities on phytopathogenic fungi被引量:3收藏 分享
作者:Zhang, Man Ru, Yifan Wang, Shilin Fu, Wen Li, Tianyu Shao, Xusheng Li, Zhong Yang, Wu-Lin
机构:East China Univ Sci & Technol;East China Univ Sci & Technol
来源:ORGANIC CHEMISTRY FRONTIERS  2024
关键词:Fungi - Iridium - Iridium compounds - Lead compounds  
质疑
Carbonyl-bridged trifluoromethyl pyridine derivatives for pest control and mechanistic investigations被引量:3收藏 分享
作者:Sheng, Zhubo Deng, Jie Yuan, Qinglong Fu, Wen Xu, Zhiping Li, Xiaoyan Li, Zhong Shao, Xusheng
机构:East China Univ Sci & Technol;East China Univ Sci & Technol;East China Univ Sci & Technol;East China Univ Sci & Technol;Guizhou Univ
来源:ADVANCED AGROCHEM  2026
关键词:TFMP   Carbonyl-bridged   Structure-activity relationships   Molecular docking   Calcium ion  
质疑
O-nitrobenzyl Caged Molecule Enables Photo-controlled Release of Thiabendazole被引量:3收藏 分享
作者:Fu, Wen Shao, Zhongli Xu, Zhiping Li, Zhong Shao, Xusheng
机构:East China Univ Sci & Technol;East China Univ Sci & Technol;East China Univ Sci & Technol;East China Univ Sci & Technol
来源:CHEMBIOCHEM  2024
关键词:Photo-controlled release   O-nitrobenzyl   Thiabendazole   Fungicidal activity   Micromorphology  
质疑
Design, Synthesis, Bioactivity, and Tentative Exploration of Action Mode for Benzyl Ester-Containing Derivatives被引量:3收藏 分享
作者:Yuan, Qinglong Fu, Wen Li, Xiaoyan Xu, Zhiping Liu, Xili Li, Zhong Shao, Xusheng
机构:East China Univ Sci & Technol;China Agr Univ;Northwest A&F Univ;China Agr Univ;East China Univ Sci & Technol
来源:JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY  2024
关键词:benzyl ester   antifungal activity   active splicing   structure-activity relationships   action mode  
质疑
N-Difluoromethylthiophthalimide Reagents for Modular Synthesis of Diversified α-Difluoromethylthiolated Ketones被引量:2收藏 分享
作者:Liang, Junqing Fu, Wen Dong, Lefeng Zhou, Cong Yuan, Qinglong Chang, Wenning Yang, Wu-Lin Xu, Xiaoyong Shao, Xusheng Li, Zhong
机构:East China Univ Sci & Technol;East China Univ Sci & Technol
来源:ORGANIC LETTERS  2023
质疑
A Terminal ModificationStrategy for Enhancing theDifference in Photoregulated Activity of Azobenzene-TolfenpyradHybrids被引量:0收藏 分享
作者:Zhang, Yongchao Qiao, Zhi Zhou, Cuncun Yin, Qi Shi, Lei Li, Zhong Fu, Wen Shao, Xusheng
机构:East China Univ Sci & Technol;Yantai Lannacheng Biotechnol Co Ltd;East China Univ Sci & Technol;Hangzhou Sinotek Qual & Technol Serv Co Ltd;East China Univ Sci & Technol
来源:JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY  2026
关键词:photopharmacology   tolfenpyrad   photochromicligand   azobenzene   photoinduced activity enhancement   photoinduced activity reduction  
质疑
Carbonyl-bridged trifluoromethyl pyridine derivatives for pest control and mechanistic investigations被引量:0收藏 分享
作者:Zhubo Sheng Jie Deng Qinglong Yuan Wen Fu Zhiping Xu Xiaoyan Li Zhong Li Xusheng Shao
机构:Shanghai Key Laboratory of Chemical Biology;State Key Laboratory of Bioreactor Engineering;Shanghai Frontier Science Research Base of Optogenetic Techniques for Cell Metabolism;Engineering Research Center of Pharmaceutical Process Chemistry;National Key Laboratory of Green Pesticide
来源:现代农业化学(英文)  2026
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Sustained-Release and Rapid-Release of Fenhexamid via the Two Different Photocages in a Light-Controllable Manner被引量:0收藏 分享
作者:Yin, Qi Li, Zongying Shao, Zhongli He, Zetao Lv, Junjie Shao, Xiaoguang Shi, Lei Fu, Wen Shao, Xusheng
机构:East China Univ Sci & Technol;Shandong Univ;Agr Comprehens Serv Ctr Xiaqiu Town;Hangzhou Sinotek Qual & Technol Serv Co Ltd;Guizhou Univ
来源:ACS AGRICULTURAL SCIENCE & TECHNOLOGY  2026
关键词:release   controllable   photocage   pesticide efficacy   fenhexamid  
质疑
Application of photopharmacology in agrochemicals被引量:0收藏 分享
作者:Wen Fu Zhong Li Xusheng Shao
机构:Shanghai Key Laboratory of Chemical Biology;State Key Laboratory of Bioreactor Engineering;Shanghai Frontier Science Research Base of Optogenetic Techniques for Cell Metabolism;Engineering Research Center of Pharmaceutical Process Chemistry
来源:现代农业化学(英文)  2023
下载全文在线阅读质疑
基于氯虫苯甲酰胺结构的PROTACs分子设计、合成及杀虫活性研究被引量:0收藏 分享
作者:张振国 付稳 李忠 邵旭升
机构:华东理工大学药学院
来源:《农药学学报》  2025
关键词:蛋白降解靶向嵌合体  鱼尼丁受体  氯虫苯甲酰胺  泊马度胺  结构改造  杀虫活性  
摘要:蛋白降解靶向嵌合体(proteolysis-targeting chimeras,PROTACs)技术作为生物医药前沿技术,可通过“事件驱动”(event driven)降解模式,特异性清除靶蛋白,因其高选择性和独特机制...
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The photoswitchable ABAMIs for the future regulation of GWT1 in a spatiotemporal level被引量:0收藏 分享
作者:Ding, Qian Li, Zongying Xiao, Zaiwei Zhang, Siting Liu, Zimai Shao, Xiaoguang Li, Zhong Fu, Wen Shao, Xusheng
机构:East China Univ Sci & Technol;Shandong Univ;Agr Comprehens Serv Ctr Xiaqiu Town;East China Univ Sci & Technol;Guizhou Univ
来源:SMART MOLECULES  2026
关键词:azobenzene-aminopyridine   bioactivity   GWT1   pesticide discovery   photoswitchable  
质疑
Wavelength-tunable light regulates binding affinity of histone deacetylase inhibitors via azobenzene Photoswitches被引量:0收藏 分享
作者:Ru, Yifan Guo, Sifan He, Yu Huang, Xiujuan Zhang, Zhenguo Shi, Lei Shao, Xiaoguang Li, Zhong Fu, Wen Shao, Xusheng
机构:East China Univ Sci & Technol;East China Univ Sci & Technol;East China Univ Sci & Technol;East China Univ Sci & Technol;Hangzhou Sinotek Qual & Technol Serv Co Ltd
来源:PESTICIDE BIOCHEMISTRY AND PHYSIOLOGY  2026
关键词:Photopharmacology   Azobenzene   Regulation   Trifluoromethyloxadiazole   HDAC   Enzymatic assay  
质疑
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