成果/Result
- Interplay of Direct Stereocontrol and Dynamic Kinetic Resolution in a Bifunctional Amine Thiourea Catalyzed Highly Enantioselective Cascade Michael-Michael Reaction被引量：69收藏
- 作者：Yu, Chenguang Zhang, Yinan Song, Aiguo Ji, Yafei Wang, Wei
- 机构：Univ New Mexico;Beijing Univ Chem Technol;E China Univ Sci & Technol;Chinese Acad Sci
- 来源：CHEMISTRY-A EUROPEAN JOURNAL 2011
- 关键词：amine thioureas cascade catalysis dynamic kinetic resolution organocatalysis tetrahydrothiophenes
- Metal-free directed C-H borylation of 2-(N-methylanilino)-5-fluoropyridines and 2-benzyl-5-fluoropyridines被引量：60收藏
- 作者：Wu, Gaorong Xu, Xiaobo Wang, Shuai Chen, Lu Pang, Binghan Ma, Tao Ji, Yafei
- 机构：East China Univ Sci & Technol;East China Univ Sci & Technol;Beijing Univ Chinese Med
- 来源：CHINESE CHEMICAL LETTERS 2022
- 关键词：Metal-free C-H borylation 2-(N-Methylanilino)-5-fluoropyridines 2-Benzyl-5-fluoropyridines BBr3
- Diastereo- and Enantioselective Organocatalytic Direct Conjugate Addition of γ-Butenolide to Chalcones被引量：56收藏
- 作者：Zhang, Yinan Yu, Chenguang Ji, Yafei Wang, Wei
- 机构：E China Univ Sci & Technol;Univ New Mexico;Chinese Acad Sci
- 来源：CHEMISTRY-AN ASIAN JOURNAL 2010
- 关键词：enones lactones Michael addition organocatalysis thioureas
- Cu(OAc)2-catalyzed remote benzylic C(sp3)-H oxyfunctionalization for C=O formation directed by the hindered para-hydroxyl group with ambient air as the terminal oxidant under ligand- and additive-free conditions被引量：44收藏
- 作者：Jiang, Jian-An Chen, Cheng Huang, Jian-Gang Liu, Hong-Wei Cao, Song Ji, Ya-Fei
- 机构：E China Univ Sci & Technol
- 来源：GREEN CHEMISTRY 2014
- Concurrent synthesis of vanillin and isovanillin被引量：42收藏
- 作者：Huang, Wei-Bin Du, Cai-Yan Jiang, Jian-An Ji, Ya-Fei
- 机构：E China Univ Sci & Technol
- 来源：RESEARCH ON CHEMICAL INTERMEDIATES 2013
- 关键词：Concurrent synthesis Vanillin Isovanillin Vilsmeier-Haack reaction Selective dealkylation
- Tandem C-C/C-N Formation via Palladium-Catalyzed C-H Activation/Styrenation and Sequential Annulation of O-Methylketoxime with Styrenes被引量：42收藏
- 作者：Fu, Xiaopan Yang, Jinyue Deng, Kezuan Shao, Lingyan Xia, Chengcai Ji, Yafei
- 机构：East China Univ Sci & Technol;Shandong First Med Univ & Shandong Acad Med Sci
- 来源：ORGANIC LETTERS 2019
- A highly efficient approach to vanillin starting from 4-cresol被引量：41收藏
- 作者：Jiang, Jian-An Chen, Cheng Guo, Ying Liao, Dao-Hua Pan, Xian-Dao Ji, Ya-Fei
- 机构：E China Univ Sci & Technol;Chinese Acad Med Sci;Peking Union Med Coll
- 来源：GREEN CHEMISTRY 2014
- C-H Borylation of Diphenylamines through Adamantane-1-carbonyl Auxiliary by BBr3被引量：29收藏
- 作者：Wu, Gaorong Fu, Xiaopan Wang, Yangyang Deng, Kezuan Zhang, Lili Ma, Tao Ji, Yafei
- 机构：East China Univ Sci & Technol;East China Univ Sci & Technol;Beijing Univ Chinese Med
- 来源：ORGANIC LETTERS 2020
- 'One-pot' synthesis of 4-substituted 1,5-diaryl-1H-pyrazole-3-carboxylates via lithium tert-butoxide-mediated sterically hindered Claisen condensation and Knorr reaction被引量：28收藏
- 作者：Jiang, Jian-An Huang, Wei-Bin Zhai, Jiao-Jiao Liu, Hong-Wei Cai, Qi Xu, Liu-Xin Wang, Wei Ji, Ya-Fei
- 机构：E China Univ Sci & Technol;Univ New Mexico
- 来源：TETRAHEDRON 2013
- 关键词：Lithium tert-butoxide Sterically hindered Claisen condensation 3-Substituted 4-aryl-2,4-diketoesters Knorr reaction 4-Substituted 1,5-diaryl-1H-pyrazole-3-carboxylates
- Practical Cu(OAc)2/TEMPO-catalyzed selective aerobic alcohol oxidation under ambient conditions in aqueous acetonitrile被引量：27收藏
- 作者：Jiang, Jian-An Du, Jia-Lei Wang, Zhan-Guo Zhang, Zhong-Nan Xu, Xi Zheng, Gan-Lin Ji, Ya-Fei
- 机构：E China Univ Sci & Technol;Roche R&D Ctr China Ltd
- 来源：TETRAHEDRON LETTERS 2014
- 关键词：Aerobic alcohol oxidation Ambient conditions Copper(II) acetate TEMPO Formation of carbonyl group
- ALTERNATE SYNTHESIS OF APIXABAN (BMS-562247), AN INHIBITOR OF BLOOD COAGULATION FACTOR XA被引量：26收藏
- 作者：Jiang, Jian'an Ji, Yafei
- 机构：E China Univ Sci & Technol
- 来源：SYNTHETIC COMMUNICATIONS 2013
- 关键词：Apixaban cost-effective synthetic route inhibitor of blood coagulation factor Xa 4-nitroaniline
- Metal-Free ortho-Selective C-H Borylation of 2-Phenylthiopyridines Using BBr3被引量：22收藏
- 作者：Wu, Gaorong Pang, Binghan Wang, Yangyang Yan, Li Chen, Lu Ma, Tao Ji, Yafei
- 机构：East China Univ Sci & Technol;East China Univ Sci & Technol;Beijing Inst Technol;Beijing Univ Chinese Med
- 来源：JOURNAL OF ORGANIC CHEMISTRY 2021
- 关键词：Reaction intermediates - Boron
- Adamantane-1-Carbonyl-Directed C-H Borylation and Hydroxylation of Benzenethiols被引量：21收藏
- 作者：Xu, Xiaobo Wu, Gaorong Yang, Zhaoziyuan Liu, Xian Hao, Liqiang Wang, Yangyang Ma, Zhihong Ji, Yafei
- 机构：East China Univ Sci & Technol;East China Univ Sci & Technol;Biotalk Co LTD
- 来源：ORGANIC LETTERS 2022
- Ruthenium(II)-Catalyzed α-Fluoroalkenylation of Oxime Ethers with gem-Difluorostyrenes via C-H Activation and C-F Cleavage被引量：21收藏
- 作者：Zhang, Lili Deng, Kezuan Wu, Gaorong Yang, Jinyue Tang, Shibiao Fu, Xiaopan Xia, Chengcai Ji, Yafei
- 机构：East China Univ Sci & Technol;Shandong First Med Univ & Shandong Acad Med Sci
- 来源：JOURNAL OF ORGANIC CHEMISTRY 2020
- 关键词：Catalysis - Ketones - Reaction intermediates - Ruthenium compounds - Activation analysis - Ethers
- Metal-Free Boron-Mediated ortho-C-H Hydroxylation of N-Benzyl-3,4,5-tribromopyrazoles被引量：19收藏
- 作者：Wu, Gaorong Yang, Zhaoziyuan Xu, Xiaobo Hao, Liqiang Chen, Lu Wang, Yangyang Ji, Yafei
- 机构：East China Univ Sci & Technol
- 来源：ORGANIC LETTERS 2022
- Efficient Co(OAc)2-catalyzed aerobic oxidation of EWG-substituted 4-cresols to access 4-hydroxybenzaldehydes被引量：18收藏
- 作者：Jiang, Jian-An Du, Jia-Lei Liao, Dao-Hua Wang, Zhan-Guo Ji, Ya-Fei
- 机构：E China Univ Sci & Technol;Roche R&D Ctr China Ltd
- 来源：TETRAHEDRON LETTERS 2014
- 关键词：Aerobic oxidation 4-Cresols 4-Hydroxybenzaldehydes Co(OAc)(2) Ethylene glycol
- Cascade Reaction for the Synthesis of Carbolines from O-Methylketoximes and Styrenes via Palladium-Catalyzed C-H Activation and Sequential Annulation被引量：18收藏
- 作者：Fu, Xiao-Pan Tang, Shi-Biao Yang, Jin-Yue Zhang, Li-Li Xia, Cheng-Cai Ji, Ya-Fei
- 机构：East China Univ Sci & Technol;Shandong First Med Univ & Shandong Acad Med Sci
- 来源：EUROPEAN JOURNAL OF ORGANIC CHEMISTRY 2019
- 关键词：Carbolines Dual C-C C-N formation Annulation Styrenes Palladium
- Palladium-Catalyzed Divergent Regioselective Homocoupling and Hydroxylation of 3-Arylbenzo[d]isoxazoles被引量：18收藏
- 作者：Guo, Ying Yu, Kun-Kun Xing, Li-Hao Liu, Hong-Wei Wang, Wei Ji, Ya-Fei
- 机构：East China Univ Sci & Technol;Univ New Mexico
- 来源：ADVANCED SYNTHESIS & CATALYSIS 2017
- 关键词：benzoisoxazoles C-H bond activation divergent synthesis homocoupling hydroxylation
- One-Pot Synthesis of 4-Substituted 1,5-Diaryl-1H-pyrazole-3-carboxylic Acids via a MeONa/LiCl-Mediated Sterically Hindered Claisen Condensation-Knorr Reaction-Hydrolysis Sequence被引量：17收藏
- 作者：Jiang, Jian-An Du, Cai-Yan Gu, Chun-Hui Ji, Ya-Fei
- 机构：E China Univ Sci & Technol
- 来源：SYNLETT 2012
- 关键词：MeONa/LiCl sterically hindered Claisen condensation Knorr reaction 4-substituted 1,5-diaryl-1H-pyrazole-3-carboxylic acids "one-pot" synthesis
- Pd-catalyzed direct oxidative mono-aroyloxylation of O-aralkyl substituted acetoxime ethers被引量：16收藏
- 作者：Shao, Ling-Yan Li, Chao Guo, Ying Yu, Kun-Kun Zhao, Fei-Yi Qiao, Wen-Li Liu, Hong-Wei Liao, Dao-Hua Ji, Ya-Fei
- 机构：East China Univ Sci & Technol;Roche R&D Ctr China Ltd
- 来源：RSC ADVANCES 2016
- 关键词：Aromatic compounds - Catalysis - Organometallics
- Pd-Catalyzed Late-Stage Monoacetoxylation and Monoiodination of 4-Alkyl-1,5-diaryl-1H-pyrazole-3-carboxylates via Direct Csp2-H Bond Activation被引量：15收藏
- 作者：Fan, Xue-Min Guo, Ying Li, Yu-Dan Yu, Kun-Kun Liu, Hong-Wei Liao, Dao-Hua Ji, Ya-Fei
- 机构：E China Univ Sci & Technol
- 来源：ASIAN JOURNAL OF ORGANIC CHEMISTRY 2016
- 关键词：acetoxylation C-H activation iodination palladium pyrazoles
- Electrochemically Induced Desulfurization of Thioureas for the Synthesis of Substituted 5-Aminotetrazoles被引量：15收藏
- 作者：Yu, Xiao Hao, Liqiang Liu, Xian Jin, Shengkui Liu, Yiping Ji, Yafei
- 机构：Minist Educ;East China Univ Sci & Technol;Chongqing Med & Pharmaceut Coll
- 来源：ADVANCED SYNTHESIS & CATALYSIS 2024
- 关键词：Addition-cyclization Desulfurization Electrosynthesis Substituted 5-aminotetrazoles
- Palladium-Catalyzed (3+2) Annulation of Aromatic Acids by C(sp3)-H Olefination and Decarboxylative Cross-Coupling Reaction被引量：15收藏
- 作者：Xu, Xiaobo Wang, Yangyang Yu, Xiao Liu, Xian Hao, Liqiang Ji, Yafei
- 机构：East China Univ Sci & Technol;East China Univ Sci & Technol
- 来源：ORGANIC LETTERS 2024
- Azobenzene-isoxazoline as photopharmacological ligand for optical control of insect GABA receptor and behavior被引量：15收藏
- 作者：Qiao, Zhi Ji, Yunfan Zhang, Yongchao Li, Zhong Xu, Zhiping Shao, Xusheng
- 机构：East China Univ Sci & Technol;East China Univ Sci & Technol
- 来源：PEST MANAGEMENT SCIENCE 2022
- 关键词：photopharmacology photochromic GABARs isoxazoline invertebrates
- Practical Ligand-Free Copper-Catalysed Short-Chain Alkoxylation of Unactivated Aryl Bromides被引量：15收藏
- 作者：Guo, Ying Fan, Xue-Min Nie, Min Liu, Hong-Wei Liao, Dao-Hua Pan, Xian-Dao Ji, Ya-Fei
- 机构：E China Univ Sci & Technol;Chinese Acad Med Sci;Peking Union Med Coll
- 来源：EUROPEAN JOURNAL OF ORGANIC CHEMISTRY 2015
- 关键词：Homogeneous catalysis Copper Alkoxylation Aromatic substitution
- Rhodium(iii)-catalyzed cascade C-H functionalization/annulation of sulfoximines with iodonium ylides for the synthesis of cyclohexanone-1,2-benzothiazines被引量：13收藏
- 作者：Chen, Lu Wang, Zhichao Wang, Yangyang Hao, Liqiang Xu, Xiaobo Wu, Gaorong Ji, Yafei
- 机构：East China Univ Sci & Technol; East China Univ Sci & Technol
- 来源：ORGANIC & BIOMOLECULAR CHEMISTRY 2022
- 关键词：Rhodium compounds - Activation analysis - Catalysis
- C-H Borylation of Benzophenones Using Hydrazone as the Traceless Directing Group被引量：13收藏
- 作者：Yang, Zhaoziyuan Hao, Liqiang Xu, Xiaobo Wang, Yangyang Wu, Gaorong Ji, Yafei
- 机构：East China Univ Sci & Technol;East China Univ Sci & Technol;Gannan Med Univ
- 来源：ORGANIC LETTERS 2023
- Rhodium(iii)-catalyzed C4-amidation of indole-oximes with dioxazolonesviaC-H activation被引量：12收藏
- 作者：Tang, Shi-Biao Fu, Xiao-Pan Wu, Gao-Rong Zhang, Li-Li Deng, Ke-Zuan Yang, Jin-Yue Xia, Cheng-Cai Ji, Ya-Fei
- 机构：East China Univ Sci & Technol;Shandong First Med Univ & Shandong Acad Med Sci
- 来源：ORGANIC & BIOMOLECULAR CHEMISTRY 2020
- 关键词：Activation analysis - Polycyclic aromatic hydrocarbons - Rhodium compounds
- Palladium-catalyzed late-stage mono-aroylation of the fully substituted pyrazoles via aromatic C-H bond activation被引量：11收藏
- 作者：Chen, Miao-Miao Shao, Ling-Yan Lun, Li Jun Wu, Yu-Liang Fu, Xiao-Pan Ji, Ya-Fei
- 机构：East China Univ Sci & Technol;Shandong Keyuan Pharmaceut Co Ltd
- 来源：CHINESE CHEMICAL LETTERS 2019
- 关键词：Palladium-catalysis Late-stage functionalization AroYlation Fully substituted pyrazoles C-H bond activation Cyclopalladated intermediate
- An Efficient One-pot Synthesis of Aryl-substituted 1-(Thiazol-2-yl)-1H-pyrazole-3-carboxylates via a Hantzsch Synthesis-Knorr Reaction Sequence被引量：11收藏
- 作者：Gu, Chunhui Zhai, Jiaojiao Jiang, Jianan Liu, Hongwei Wang, Lei Zhu, Dunru Ji, Yafei
- 机构：E China Univ Sci & Technol;Nanjing Univ Technol
- 来源：CHINESE JOURNAL OF CHEMISTRY 2014
- 关键词：one-pot synthesis Claisen condensation Hantzsch synthesis Knorr reaction 1-(thiazol-2-yl)pyrazole-3-carboxylates
